Table 2 Percentage of incorporation of 213BiIII by chelate ligands (pH 5.5, V = 0.1 mL, reaction time 5 min at 95 °C). Data represent mean values ± SD, n = 3
c [μM] | DOTP | DOTPH | DOTPOEt | DOTPI | CHX-A"-DTPA | DOTA |
|---|---|---|---|---|---|---|
100 | 99.4 ± 0.3 | 98.7 ± 2.1 | 99.1 ± 0.1 | 99.7 ± 0.3 | 99.8 ± 0.1 | 96.9 ± 3.6 |
30 | 98.6 ± 0.9 | 99.0 ± 0.2 | 99.0 ± 1.0 | 98.8 ± 0.3 | 96.8 ± 2.4 | 94.3 ± 2.6 |
10 | 96.4 ± 2.3 | 99.1 ± 0.7 | 98.3 ± 0.9 | 94.2 ± 4.2 | 91.9 ± 1.9 | 81.1 ± 9.0 |
3 | 94.3 ± 2.1 | 92.7 ± 2.5 | 96.4 ± 0.6 | 92.9 ± 4.8 | 89.2 ± 6.9 | 64.1 ± 21.4 |
1 | 91.8 ± 4.0 | 85.4 ± 2.6 | 95.9 ± 0.3 | 88.0 ± 10.8 | 90.2 ± 6.6 | 37.4 ± 17.5 |
0.3 | 90.6 ± 3.9 | 79.7 ± 4.7 | 94.7 ± 0.7 | 73.6 ± 29.0 | 82.7 ± 5.3 | 14.6 ± 6.1 |
0.1 | 90.9 ± 3.2 | 79.0 ± 2.5 | 93.7 ± 2.6 | 31.7 ± 17.1 | 49.7 ± 23.1 | 3.8 ± 2.8 |
0.03 | 90.4 ± 4.5 | 72.0 ± 5.4 | 85.7 ± 3.9 | 20.2 ± 9.4 | 9.8 ± 9.2 | |
0.01 | 89.5 ± 1.0 | 61.8 ± 8.7 | 66.2 ± 5.8 | 6.5 ± 4.7 | ||
0.003 | 56.2 ± 6.1 | 37.3 ± 5.5 | 10.5 ± 3.7 | |||
0.001 | 5.3 ± 4.2 | 0.4 ± 0.6 | 2.5 ± 0.7 |