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Table 1 NOTA/NODA ligands and maximum isolated yields after radiolabeling with 500 nmol peptide ( R = K d (HSG)Y d K d (HSG)-NH 2 )

From: Radiofluorination using aluminum-fluoride (Al18F)

Peptide

Structure

Maximum 18F-labeling yield (%)

IMP449

44

IMP460

5.8

IMP461

31

IMP467

87

  1. Reproduced with permission from Bioconjugate Chemistry, McBride et al. [23].