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Table 3 Transmetallation of [68Ga]Ga-4HMSA in presence of various biologically relevant metal salts

From: [68Ga]Ga-4HMSA a promising new PET tracer for imaging inflammation

Metal (10 equiv)

% of Remaining Ga68 complexation

15 min

30 min

60 min

CoCl2

100a

100b

100a

100b

100a

100b

CuCl2

100a

100b

100a

100b

78a

95b

FeCl3

100a

100b

71a

86b

35a

72b

NiCl2

100a

100b

100a

100b

100a

100b

MgCl2

100a

100b

100a

100b

100a

100b

  1. apH = 2.0; bpH = 7.4