From: Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
Compounds
KD at the hY1R (nM)
[F7,P34]-NPY
0.94 ± 0.08
pb12
3.1 ± 0.8
[111In]In-pb12
5.1 ± 3.5
[natTb]Tb-pb12
30 ± 3.7
pb13
No specific binding
[111In]In-pb13
[natTb]Tb-pb13