Skip to main content

Table 1 Numerical values of the SPECT and metabolite protocol parameters corresponding to the 18 experiments

From: In vivo absolute quantification of striatal and extrastriatal D2/3 receptors with [123I]epidepride SPECT

Rats

Modality/tracer

Duration (min)

Injection 1 (T = 0 min)

Injection 2

Injection 3

SA† (GBq/μmol)

J1* (MBq/μg)

Time (min)

J2* (MBq/μg)

J2 (μg)

Time (min)

J3 (μg)

1

TLC/[123I]epidepride

180

> 1000

89.6/< 0.05

–

–

–

–

–

2

TLC/[123I]epidepride

180

> 1000

98.2/< 0.05

–

–

–

–

–

3

TLC/[123I]epidepride

180

> 1000

96.9/< 0.05

–

–

–

–

–

4

TLC/[123I]epidepride

180

> 1000

77.4/< 0.05

–

–

–

–

–

5

SPECT-MI/[123I]epidepride

360

1065.86

95.4/0.043

180

103.4/0.047

1.07

240

214.00

6

SPECT-MI/[123I]epidepride

360

967.71

87.4/0.043

180

93.5/0.046

2.35

240

234.50

7

SPECT-MI/[123I]epidepride

360

955.45

87.6/0.044

180

97.5/0.049

1.10

240

221.00

8

SPECT-PSA/[123I]epidepride

180

19.50

52.7/1.30

–

–

–

–

–

9

SPECT-PSA/[123I]epidepride

180

23.74

58.6/1.19

–

–

–

–

–

10

SPECT-PSA/[123I]epidepride

180

40.67

113.06/1.34

–

–

–

–

–

11

SPECT-PSA/[123I]epidepride

180

29.51

75.24/1.23

–

–

–

–

–

12

SPECT-PSA_CON/[123I]epidepride

180

18.85

49.35/1.26

–

–

–

–

–

13

SPECT-PSA_CON/[123I]epidepride

180

16.98

43.48/1.23

–

–

–

–

–

14

SPECT-PSA_CON/[123I]epidepride

180

22.74

45.65/0.97

–

–

–

–

–

15

SPECT-PSA_CON/[123I]epidepride

180

17.10

41.15/1.16

–

–

–

–

–

16

SPECT-PSA_HAL/[123I]epidepride

180

18.81

46.09/1.18

–

–

–

–

–

17

SPECT-PSA_HAL/[123I]epidepride

180

16.72

40.7/1.17

–

–

–

–

–

18

SPECT-PSA_HAL/[123I]epidepride

180

16.95

38.47/1.09

–

–

–

–

–