From: [111In]PSMA-I&T: expanding the spectrum of PSMA-I&T applications towards SPECT and radioguided surgery
Ligand
IC50 [nM]
Internalization [% of reference]
Lipophilicity [log POW]
In-PSMA-I&T
7.5 ± 1.5
104 ± 7
−4.5
Ga-PSMA-I&T
9.4 ± 2.9
59 ± 2
−4.3
Lu-PSMA-I&T
7.9 ± 2.4
76 ± 2
−4.1