n ≥ 3 | [11C]Me@HAPTHI | |
---|---|---|
% BL-competitor | fmol | |
Rat heart | ||
 FMeNER 1 μM | 88.8 ± 11.2 | <0.01 |
 FMeNER 100nM | 99.00 ± 0.07 | <0.01 |
 Me@HAPTHI 1 μM | 92.5 ± 7.5* | <0.01 |
 Me@HAPTHI 100nM | 104.5 ± 4.5 | <0.01 |
Human cortex | ||
 FMeNER 1 μM | 71.9 ± 7.9* | 0.86 |
 FMeNER 100nM | 86.3 ± 11.2* | <0.01 |
 Me@HAPTHI 1 μM | 66.3 ± 5.9* | 1.32 |
 Me@HAPTHI 100nM | 82.1 ± 13.9* | 0.02 |
Human thalamus | ||
 FMeNER 1 μM | 68.36 ± 2.11 | 0.71 |
 FMeNER 100nM | 77.6 ± 9.8 | 0.47 |
 Me@HAPTHI 1 μM | 85.9 ± 18.5 | 0.09 |
 Me@HAPTHI 100nM | 92.5 ± 17.3 | 0.26 |
Human hypothalamus | ||
 FMeNER 1 μM | 77.4 ± 14.5 | 0.02 |
 FMeNER 100 nM | 97.8 ± 14.6 | 0.11 |
 Me@HAPTHI 1 μM | 62.0 ± 3.6* | 0.04 |
 Me@HAPTHI 100 nM | 83.7 ± 1.7* | 0.05 |
Human hippocampus | ||
 FMeNER 1 μM | 67.3 ± 8.2 | <0.01 |
 FMeNER 100 nM | 97.1 ± 10.3 | <0.01 |
 Me@HAPTHI 1 μM | 68.3 ± 5.3 | <0.01 |
 Me@HAPTHI 100 nM | 84.1 ± 9.3 | <0.01 |
Human nucleus caudatus | Â | Â |
 FMeNER 1 μM | 107.6 ± 17.7 | n.d. |
 FMeNER 100nM | 102.6 ± 14.5 | n.d. |
 Me@HAPTHI 1 μM | 110.0 ± 21.0 | n.d. |
 Me@HAPTHI 100nM | 93.5 ± 12.5 | nd |
Human cerebellum | Â | Â |
 FMeNER 1 μM | 108.2 ± 17.3 | n.d. |
 FMeNER 100nM | 103.9 ± 12.2 | n.d. |
 Me@HAPTHI 1 μM | 107.2 ± 20.8 | n.d. |
 Me@HAPTHI 100nM | 124.7 ± 10.8 | n.d. |