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Table 4 Tissue exposure (AUC) for the duration of the PET scan

From: Lapatinib access into normal brain and brain metastases in patients with Her-2 overexpressing breast cancer

Normal brain

AUC (min.g/mL)

Tumour metastases

AUC (min.g/mL)

Sub 1 - BL

319.6318

Sub 4 met - BL

708.198

Sub 1 - D 8

328.7575

Sub 4 met - D 8

623.23

Sub 3 - BL

304.0247

Sub 7 met 1 - BL

518.227

Sub 3 - D 8

301.1074

Sub 7 met 1 - D 8

665.909

Sub 4 - BL

203.6962

Sub 7 met 2 - BL

2,584.31

Sub 4 - D 8

198.8753

Sub 7 met 2 - D 8

2,757.86

Sub 7 - BL

289.1109

Sub 10 met 1 - D 8

2,731.19

Sub 7 - D 8

272.9378

Sub 10 met 2 - D 8

1,577.81

Sub 9 - D 8

233.2629

Sub 10 met 3 - D 8

2,289.3

Sub 10 - D 8

252.7335

Sub 10 met 4 - D 8

1,647.02

  1. AUC, area under the curve concentration; BL, baseline; D, day; met, metastases; min, minutes; PET, positron emission tomography; Sub, subject.