|
11C-LY2428703
|
18F-FMPEP
[22]
|
18F-SP203
[19]
|
11C-( R)-rolipram
[23]
|
11C-NOP1A
[24]
|
---|
Target
|
mGluR1
|
CB1
|
mGluR5
|
PDE4
|
NOP
|
Brain peak SUV
|
~0.5
|
3 to 4
|
~6
|
2 to 2.5
|
5 to 7
|
Exposure SUV (0 to 20)
|
202.2
|
47.8
|
37.0
|
124.9
|
36.7
|
f
p %
|
0.094
|
0.63
|
5.2
|
6.4
|
10.1
|
Effective exposure (E × f
p)
|
0.19
|
0.30
|
1.9
|
8.0
|
3.7
|