Peptide | [M] + | Yield | Purity b | Ki c | Labeling | |
---|---|---|---|---|---|---|
Calcd | Found a | (%) | (%) | (nM) | yield d (%) | |
Bombesin | 0.59 ± 0.32 | |||||
NOTA-monomer | 1,570 | 1,571 | 38 | 99 | 2.51 ± 1.54e | > 95 |
South BBN peptide segment | 1,879 | 1,880 | 84f | |||
NOTA-dimer 1 | 2,976 | 2,976 | 28 | 99 | 2.00 ± 1.59 | > 95 |
NOTA-dimer 2 | 3,122 | 3,122 | 31 | 99 | 1.76 ± 1.30 | > 95 |