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Table 1 Overview of [ 11 C]phenytoin scans

From: [11C]phenytoin revisited: synthesis by [11C]CO carbonylation and first evaluation as a P-gp tracer in rats

Animal

Scan 1

Scan 2

Scan 3

1

Baseline

-

-

2

Baseline

-

-

3

Baseline

Tariquidar 15 mg·kg−1

-

4

Tariquidar 15 mg·kg−1

Tariquidar 15 mg·kg−1

-

5

Baseline

Probenecid 150 mg·kg−1

Tariquidar 15 mg·kg−1

6

Baseline

Probenecid 150 mg·kg−1

Tariquidar 15 mg·kg−1